6-溴呋喃并[3,2-b]吡啶合成路线 (共 1 条)
反应条件
sodium carbonate; tetrakis(triphenylphosphine) palladium(0) in water; N,N-dimethyl-formamide T=120°C; 2 h; Microwave irradiation;
参考文献
NOVARTIS AG; BETSCHART, Claudia; COTESTA, Simona; HINTERMANN, Samuel; WAGNER, Juergen; ROY, Bernard, Lucien; GERSPACHER, Marc; VON MATT, Anette; BEHNKE, Dirk
Patent: WO2011/73316 A1, 2011 ;
Location in patent: Page/Page column 69-70 ;
WO 2011/073316 A1