4-(2-(哌啶-1-基)乙氧基)苯基硼酸频哪醇酯合成路线 （共 2 条）
反应条件
1: 4-[4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl]-phenol With potassium carbonate in N,N-dimethyl-formamide
T=0°C;
2: N-(2-chloroethyl)-piperidine hydrochloride With tetra-(n-butyl)ammonium iodide in N,N-dimethyl-formamide
T=50°C;
参考文献
Malo-Forest, Bianca; Landelle, Gregory; Roy, Jessye-Ann; Lacroix, Jacques; Gaudreault, Rene C.; Paquin, Jean-Francois
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 6 p. 1712 - 1715
反应条件
1.1: potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride / dimethyl sulfoxide / 80 °C
2.1: potassium carbonate / N,N-dimethyl-formamide / 0 °C
2.2: 50 °C
View Scheme
参考文献
Malo-Forest, Bianca; Landelle, Gregory; Roy, Jessye-Ann; Lacroix, Jacques; Gaudreault, Rene C.; Paquin, Jean-Francois
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 6 p. 1712 - 1715
