反应条件
1: POCl3, N,N-dimethylaniline / toluene / 3 h / Heating
2: toluene / 3 h / Heating
3: EtSH, AlCl3 / 4 h / Ambient temperature
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参考文献
Liao, Yi; DeBoer, Peter; Meier, Eddie; Wikstroem, Hakan
Journal of Medicinal Chemistry, 1997 , vol. 40, # 25 p. 4146 - 4153