4-羟基甲基-7-氮杂吲哚合成路线 (共 11 条)
反应条件
1.1: trichlorophosphate / Reflux
1.2: pH 9
2.1: calcium chloride; sodium tetrahydroborate / tetrahydrofuran / 6 h / Reflux
View Scheme
参考文献
ASCEPION PHARMACEUTICALS, INC.; JIANG, Shan; XING, Xinglong; WANG, Qishan; KONG, Ren
Patent: WO2011/23081 A1, 2011 ;
WO 2011/023081 A1