1: With boron trifluoride diethyl etherate in dichloromethane T=-20°C; 0.0833333 h; 2: With water; sodium hydrogencarbonate in dichloromethane optical yield given as percent destereoselective reaction;
参考文献
Cresswell, Alexander J.; Davies, Stephen G.; Lee, James A.; Roberts, Paul M.; Russell, Angela J.; Thomson, James E.; Tyte, Melloney J.
Organic Letters, 2010 , vol. 12, # 13 p. 2936 - 2939
1: benzyl chloride With iodine; zinc in N,N-dimethyl acetamide T=80°C; 2: chloroacetyl chloride With tetrakis(triphenylphosphine) palladium(0) in N,N-dimethyl acetamide T=20°C;
参考文献
Journal of Medicinal Chemistry, , vol. 50, # 1 p. 40 - 64