7-溴吡咯并[1,2-f][1,2,4]噻嗪-4-胺合成路线 (共 2 条)
反应条件
1,3-dibromo-5,5-dimethyl-hydantoin in N,N-dimethyl-formamide T=-20°C; 1.5 h;
参考文献
BAYER PHARMACEUTICALS CORPORATION
Patent: WO2007/64931 A2, 2007 ;
Location in patent: Page/Page column 164 ;
反应条件
1: With n-butyllithium in tetrahydrofuran T=-78°C; 0.25 h; 2: With water in tetrahydrofuran
参考文献
BAYER PHARMACEUTICALS CORPORATION
Patent: WO2007/64931 A2, 2007 ;
Location in patent: Page/Page column 168 ;