4-(6-氯-嘧啶-4-基氨基)-哌啶-1-羧酸叔丁酯合成路线 (共 1 条)
反应条件
triethylamine in dichloromethane T=20°C; 72 h;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH; NEUROCRINE BIOSCIENCES, INC.; TRAN, Joe, A.; CHEN, Chen
Patent: WO2010/149685 A1, 2010 ;
Location in patent: Page/Page column 49 ;
WO 2010/149685 A1