3-(6-氯-嘧啶-4-基氨基)-哌啶-1-羧酸叔丁酯合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in butan-1-ol
T=120°C; 12 h;
参考文献
AVILA THERAPEUTICS, INC.; TESTER, Richland, W.
Patent: WO2009/51822 A1, 2009 ;
Location in patent: Page/Page column 137-138 ;
WO 2009/051822 A1