2-甲基硫代嘧啶-5-硼酸频那酯合成路线 (共 2 条)
反应条件
potassium acetate; palladium diacetate in N,N-dimethyl-formamide T=20 - 85°C; Inert atmosphere;
参考文献
WO2010/9183 A1, ;
Page/Page column 110 ;
WO 2010/009183 A1
反应条件
sodium peroxoborate tetrahydrate; water in tetrahydrofuran T=20°C; Inert atmosphere;
参考文献
BRISTOL-MYERS SQUIBB COMPANY; WACKER, Dean, A.; ROSSI, Karen, A.; WANG, Ying; WU, Gang
Patent: WO2010/9183 A1, 2010 ;
Location in patent: Page/Page column 110 ;
WO 2010/009183 A1