1,2,3,4-四氢咔唑合成路线 （共 202 条）
反应条件
sulfuric acid 1 h; Heating;
参考文献
Davis, Paul D.; Neckers, Douglas C.
Journal of Organic Chemistry, 1980 , vol. 45, # 3 p. 456 - 462
反应条件
water-d2; tert.-butyl lithium; pentane in hexane 1) - 78 deg C; 2) r.t., 16 h;
参考文献
Magnetic Resonance in Chemistry, , vol. 26, p. 347 - 350
反应条件
in pyridine; ethanol; water; cyclohexanone
反应条件
pyridine in N,N-dimethyl-formamide
参考文献
Wender, Paul A.; White, Alan W.
Tetrahedron, 1983 , vol. 39, # 22 p. 3767 - 3776
反应条件
hydrogen in tetrahydrofuran T=150°C; P=37503.8 Torr; 1 h;
参考文献
Dalton Transactions, , vol. 40, # 40 p. 10621 - 10632
反应条件
in cyclohexane 1.8 h; Irradiation;
参考文献
Wender, Paul A.; Cooper, Christopher B.
Tetrahedron, 1986 , vol. 42, # 11 p. 2985 - 2992
反应条件
hydroxyapatite-bound Pd in water T=110°C; 3 h;
参考文献
Hara, Takayoshi; Mori, Kohsuke; Mizugaki, Tomoo; Ebitani, Kohki; Kaneda, Kiyotomi
Tetrahedron Letters, 2003 , vol. 44, # 33 p. 6207 - 6210
反应条件
1: 78 percent / AgF / H2O 2: 89 percent / CO2 / dimethylsulfoxide; CH2Cl2; acetonitrile / -40 - 20 °C 3: 88 percent / aq. TiCl3; NH4OAc / acetone / 0.25 h / 20 °C View Scheme
参考文献
Organic Letters, , vol. 1, # 4 p. 673 - 676
反应条件
1: 45 percent / P(tBu)3; Cs2CO3 / Pd(OAc)2 / toluene 2: 89 percent / TsOH*H2O / toluene / 2 h / 80 °C View Scheme
参考文献
Tetrahedron Letters, , vol. 45, # 9 p. 1857 - 1859
反应条件
in hydrogenchloride; isopropyl alcohol T=20°C; Heating; MechanismKineticsThermodynamic data;
参考文献
Journal of the Chemical Society, Perkin Transactions 2: Physical Organic Chemistry (1972-1999), , p. 1215 - 1220
