反应条件
1: With lithium hydroxide hydrate; water in 1,4-dioxane
T=20°C; 1 h;
2: With citric acid in 1,4-dioxane; water
参考文献
F. HOFFMANN-LA ROCHE AG; BISSANTZ, Caterina; DEHMLOW, Henrietta; ERICKSON, Shawn David; KARNACHI, Prabha Saba; KIM, Kyungjin; MARTIN, Rainerm, E.; MATTEI, Patrizio; OBST SANDER, Ulrike; PIETRANICO-COLE, Sherrie Lynn; RICHTER, Hans; ULLMER, Christoph
Patent: WO2012/117000 A1, 2012 ;
Location in patent: Page/Page column 197 ;