反应条件
1: (S)-α,α-diphenylprolinol - n-butylboronic acid, catecholborane / toluene / 12 h / -78 °C 2: 91 percent / NaN3, NaOH, H2O / 1,2-dimethoxy-ethane / 24 h / 23 °C 3: 92 percent / H2 / 10percent Pd/C / ethyl acetate / 13 h / 760 Torr View Scheme
参考文献
Journal of the American Chemical Society, , vol. 114, # 5 p. 1906 - 1908