2-(1,2,3,6-四氢吡啶-4-基)-5-(三氟甲基)吡啶合成路线 (共 1 条)
反应条件
potassium carbonate; tetrakis(triphenylphosphine) palladium(0); dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in N,N-dimethyl-formamide
T=125°C; 0.5 h; Microwave;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2007/76318 A2, 2007 ;
Location in patent: Page/Page column 62 ;
WO 2007/076318 A2