2-甲基-1-苯磺酰基-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡咯并[2,3-B]吡啶合成路线 (共 1 条)
反应条件
potassium acetate; dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in N,N-dimethyl-formamide
T=90°C; 12 h;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2007/76423 A2, 2007 ;
Location in patent: Page/Page column 171 ;
WO 2007/076423 A2