6-溴咪唑并[1,2-a]吡啶-3-羧酸合成路线 (共 2 条)
反应条件
1: With water; lithium hydroxide hydrate in tetrahydrofuran; methanol T=60°C; 2: With hydrogenchloride in water pH=4;
参考文献
WO2011/50245 A1, ;
Page/Page column 105 ;
WO 2011/050245 A1
反应条件
1.1: ethanol / Reflux 2.1: water; lithium hydroxide hydrate / tetrahydrofuran; methanol / 60 °C 2.2: pH 4 View Scheme
参考文献
WO2011/50245 A1, ;
WO 2011/050245 A1