7-氟-3-碘-1H-吲唑合成路线 (共 1 条)
反应条件
iodine; potassium hydroxide in N,N-dimethyl-formamide
T=50°C; 0.333333 h;
参考文献
DAINIPPON SUMITOMO PHARMA CO., LTD.; MIZUNO, Kazuhiro; IKEDA, Junya; NAKAMURA, Takanori; IWATA, Masato; OTAKA, Hiromichi; GOTO, Nana
Patent: WO2012/169649 A1, 2012 ;
Location in patent: Page/Page column 192 ;
WO 2012/169649 A1