2-甲基-5-(1,3-恶唑-2-基)苯硼酸频哪醇酯合成路线 (共 1 条)
反应条件
dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct; potassium acetate in 1,4-dioxane; water
T=100°C; 48 h; Schlenk techniqueInert atmosphere;
参考文献
Almirall, S.A.; Vidal Juan, Bernat; Gonzalez Rodriguez, Jacob; Gual Roig, Silvia; Esteve Trias, Cristina; Vidal Gispert, Laura
Patent: EP2738172 A1, 2014 ;
Location in patent: Paragraph 0108; 0168 ;