7-氨基-5-氟吲哚啉-2-酮合成路线 (共 2 条)
反应条件
hydrogen; 5 Pd(II)/C(eggshell) in acetic acid
T=20°C;
参考文献
Shanghai Hengrui Pharmaceutical Co. Ltd.
Patent: EP2157093 A1, 2010 ;
Location in patent: Page/Page column 51 ;
反应条件
sulfuric acid; nitric acid
T=-5 - 20°C;
参考文献
Tang, Peng Cho; Su, Yidong; Zhang, Lei; Xiao, Lu
Patent: US2010/4239 A1, 2010 ;
Location in patent: Page/Page column 56-57 ;