1: With lithium borohydride in tetrahydrofuran
T=0 - 20°C; 48 h;
2: With water in tetrahydrofuran; ethyl acetate
参考文献
UNIVERSITY OF VIRGINIA PATENT FOUNDATION; BIOGEN IDEC MA INC.
Patent: WO2009/23854 A1, 2009 ;
Location in patent: Page/Page column 37; 41; 3/22 ;
WO 2009/023854 A1