4-(三氟甲基)吡啶-3-硼酸合成路线 (共 1 条)
反应条件
1: With n-butyllithium in tetrahydrofuran T=-78 - 20°C; Inert atmosphere; 2: With water in tetrahydrofuran
参考文献
PAMLICO PHARMACEUTICAL INC.; ATKINSON, Robert N.; OMMEN, Andy J.; VEAL, James M.; HUANG, Kenneth H.; SMITH, Emilie, D.
Patent: WO2012/88411 A1, 2012 ;
Location in patent: Page/Page column 69 ;