Annogen; sodium hydroxide; palladium dichloride in water; acetonitrile T=80°C; pH=12;
参考文献
Jagadeesh, Rajenahally V.; Sandhya, Y. Sree; Karthikeyan; Reddy, S. Sudhakar; Reddy, P. Pradeep Kumar; Kumar, M. Viniod; Charan, K. T. Prabhu; Narender; Bhagat
Synthetic Communications, 2011 , vol. 41, # 16 p. 2343 - 2349
1: cyclobenzothiazole With n-butyllithium in tetrahydrofuran T=-78°C; 0.5 h; 2: N,N-dimethyl-formamide in tetrahydrofuran T=-78 - 20°C; 2 h; 3: With water; ammonium chloride in tetrahydrofuran
参考文献
ZENOBIA THERAPEUTICS, INC.; BOUNAUD, Pierre-Yves; NIENABER, Vicki; STEENSMA, Ruo, W.; LOWE, John, A., III
Patent: WO2012/178015 A2, 2012 ;
Location in patent: Page/Page column 114 ;
WO 2012/178015 A2
