Dorofeenko,G.N. et al.
Chemistry of Heterocyclic Compounds (New York, NY, United States), 1973 , vol. 9, p. 944 - 947
Khimiya Geterotsiklicheskikh Soedinenii, 1973 , vol. 9, p. 1016 - 1019
1.1: n-BuLi / tetrahydrofuran; hexane / 1 h / -78 °C
1.2: tetrahydrofuran; hexane / 2 h / -78 °C
2.1: 10percent aq. AcOH / acetone / 2 h / Heating
View Scheme
参考文献
Wells, Geoffrey; Berry, Jane M.; Bradshaw, Tracey D.; Burger, Angelika M.; Seaton, Angela; Wang, Bo; Westwell, Andrew D.; Stevens, Malcolm F. G.
Journal of Medicinal Chemistry, 2003 , vol. 46, # 4 p. 532 - 541