Masters, Kye-Simeon; Rauws, Tom R. M.; Yadav, Ashok K.; Herrebout, Wouter A.; Van Der Veken, Benjamin; Maes, Bert U. W.
Chemistry - A European Journal, 2011 , vol. 17, # 23 p. 6315 - 6320
El-Sharief, A. M. Sh.; Hammad, N.E.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1981 , vol. 20, # 12 p. 1039 - 1042
1: pyridine / CH2Cl2 / 0 °C
2: ClSO3H / 60 °C
3: NH3 / CH2Cl2 / 20 °C
View Scheme
参考文献
Kim, Semi; Park, Ji Hyun; Koo, Sun-Young; Kim, Jung In; Kim, Min-Hyeung; Kim, Ji Eun; Jo, Kiwon; Geun Choi, Hwan; Lee, Sung Bae; Jung, Sang-Hun
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 24 p. 6075 - 6078
1: 2-acetoxy-3-bromo-5-chlorobenzoic acid With triethylamine; isobutyl chloroformate in tetrahydrofuran
T=-15°C; 0.0833333 h;
2: 2-chloro-aniline in tetrahydrofuran
T=20°C; 48 h;
参考文献
Kanamori, Daisuke; Okamura, Taka-Aki; Yamamoto, Hitoshi; Shimizu, Shigeomi; Tsujimoto, Yoshihide; Ueyama, Norikazu
Bulletin of the Chemical Society of Japan, 2004 , vol. 77, # 11 p. 2057 - 2064