1: With sodium hydrogencarbonate in tetrahydrofuran; water T=20 - 80°C; 20 h; 2: With lithium aluminium tetrahydride in tetrahydrofuran T=20°C; 2 h; 3: With water; sodium hydrogencarbonate in tetrahydrofuran
参考文献
CHEMOCENTRYX, INC.
Patent: WO2006/76644 A2, 2006 ;
Location in patent: Page/Page column 187 ;
WO 2006/076644 A2