2-氨基-4-氯苯酚合成路线

参考文献

Sharifi, Ali; Barazandeh, Mehdi; Saeed Abaee; Mirzaei, Mojtaba
Tetrahedron Letters, 2010 , vol. 51, # 14 p. 1852 - 1855

参考文献

Caliendo, Giuseppe; Grieco, Paolo; Perissutti, Elisa; Santagada, Vincenzo; Santini, Antonello; Albrizio, Stefania; Fattorusso, Caterina; Pinto, Aldo; Sorrentino, Raffaella
European Journal of Medicinal Chemistry, 1998 , vol. 33, # 12 p. 957 - 967

598-21-0溴乙酰溴+

95-85-22-氨基-4-氯苯酚

7652-29-16-氯-2H-1,4-苯并噁嗪-3(4H)-酮

参考文献

Geng, Bolin; Comita-Prevoir, Janelle; Eyermann, Charles J.; Reck, Folkert; Fisher, Stewart
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 18 p. 5432 - 5435

74974-54-22-氯-1,1,1-三甲氧基乙烷+

95-85-22-氨基-4-氯苯酚

63842-22-85-氯-2-氯甲基-1,3-苯并噁唑

参考文献

ARGENTA DISCOVERY LIMITED; ASTRAZENECA AB
Patent: WO2009/153536 A1, 2009 ;
Location in patent: Page/Page column 37-38 ;
WO 2009/153536 A1

95-85-22-氨基-4-氯苯酚

63842-22-85-氯-2-氯甲基-1,3-苯并噁唑

参考文献

Pfizer Inc.
Patent: US4723010 A1, 1988 ;

51076-95-02-氯-1,1,1-三乙氧基乙烷+

95-85-22-氨基-4-氯苯酚

63842-22-85-氯-2-氯甲基-1,3-苯并噁唑

参考文献

Mylari; Beyer; Scott; Aldinger; Dee; Siegel; Zembrowski
Journal of Medicinal Chemistry, 1992 , vol. 35, # 3 p. 457 - 465

3674-13-32,3-二溴丙酸乙酯+

95-85-22-氨基-4-氯苯酚

68281-43-66-氯-3,4-二氢-2H-苯并[1,4]噁嗪-2-羧酸乙酯

参考文献

Maingot, Lucie; Elbakali, Jamal; Dumont, Julie; Bosc, Damien; Cousaert, Nicolas; Urban, Agathe; Deglane, Gaelle; Villoutreix, Bruno; Nagase, Hideaki; Sperandio, Olivier; Leroux, Florence; Deprez, Benoit; Deprez-Poulain, Rebecca
European Journal of Medicinal Chemistry, 2013 , vol. 69, p. 244 - 261

95-85-22-氨基-4-氯苯酚

1276666-16-0+

1276666-14-8(5R)-4-(5-氯-1,3-苯并恶唑-2-基)-5-甲基-1,4-二氮杂环庚烷-1-鎓 (2S,3S)-2,3-二(苯甲酰氧基)丁二酸盐

参考文献

MERCK SHARP and DOHME CORP.; MERCK SHARP and DOHME LIMITED; BAXTER, Carl, A.; CLEATOR, Edward; KRSKA, Shane, W.; SHEEN, Faye; STEWART, Gavin; STROTMAN, Neil; WALLACE, Debra, J.; WRIGHT, Timothy
Patent: WO2012/148553 A1, 2012 ;
WO 2012/148553 A1

95-85-22-氨基-4-氯苯酚

1276666-13-75-氯-2-(六氢-5-甲基-1H-1,4-二氮杂卓-1-基)苯并恶唑

参考文献

MERCK SHARP and DOHME CORP.; MERCK SHARP and DOHME LIMITED; BAXTER, Carl, A.; CLEATOR, Edward; KRSKA, Shane, W.; SHEEN, Faye; STEWART, Gavin; STROTMAN, Neil; WALLACE, Debra, J.; WRIGHT, Timothy
Patent: WO2012/148553 A1, 2012 ;
WO 2012/148553 A1

3151-49-3+

95-85-22-氨基-4-氯苯酚

1298023-69-4

参考文献

Jadhav, Gopal P.; Chhabra, Siri Ram; Telford, Gary; Hooi, Doreen S. W.; Righetti, Karima; Williams, Paul; Kellam, Barrie; Pritchard, David I.; Fischer, Peter M.
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