1: With hydrazine in ethanol
Heating / reflux;
2: With hydrogenchloride in ethanol; water
T=50°C; 0.5 h;
3: With sodium hydroxide in ethanol; water
T=0°C; pH=10 - 12;
参考文献
PROBIODRUG AG
Patent: US2008/267912 A1, 2008 ;
Location in patent: Page/Page column 32 ;
US 20080267912 A1