甲基(2,4-二氟苯基)乙酸酯合成路线 (共 2 条)
反应条件
sulfuric acid
T=20°C; 18 h; Reflux;
参考文献
JANSSEN PHARMACEUTICALS, INC.; CID-NUNEZ, Jose, Maria; TRABANCO-SUAREZ, Andres, Avelino; VEGA RAMIRO, Juan, Antonio; OEHLRICH, Daniel; TRESADERN, Gary, John; MACDONALD, Gregor, James
Patent: WO2012/62759 A1, 2012 ;
Location in patent: Page/Page column 47 ;
WO 2012/062759 A1
反应条件
potassium carbonate in N,N-dimethyl-formamide
参考文献
Amgen Inc.
Patent: US2007/299080 A1, 2007 ;
Location in patent: Page/Page column 72 ;