4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吲哚-6-羧酰胺合成路线 (共 2 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dimethyl sulfoxide
T=90°C;
参考文献
PIRAMED LIMITED; THE INSTITUTE OF CANCER RESEARCH
Patent: WO2008/125839 A2, 2008 ;
Location in patent: Page/Page column 21; 27; 33 ;
WO 2008/125839 A2
参考文献
PIRAMED LIMITED
Patent: WO2007/122410 A1, 2007 ;
Location in patent: Page/Page column 73 ;