1: in N,N-dimethyl acetamide T=60°C; 2: With hydrogenchloride in methanol; N,N-dimethyl acetamide; water 2 h; Heating / reflux; Product distribution / selectivity;
参考文献
SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH
Patent: WO2008/119015 A2, 2008 ;
Location in patent: Page/Page column 54 ;