反应条件
1: 44 percent / POCl3; N,N-diethylaniline / 1,2-dichloro-ethane / 3 h / Heating
2: 33 percent / K2CO3 / H2O / 4 h / 120 °C
View Scheme
参考文献
Norman; Chen; Fotsch; Hale; Han; Hurt; Jenkins; Kincaid; Liu; Lu; Moreno; Santora; Sonnenberg; Karbon
Journal of Medicinal Chemistry, 2000 , vol. 43, # 22 p. 4288 - 4312