1: With hydrogen; palladium on activated charcoal in methanol T=20°C; P=3000.3 Torr; 18 h; 2: With lithium aluminium tetrahydride in tetrahydrofuran 3: With water in tetrahydrofuran
参考文献
SCHWARZ PHARMA AG
Patent: WO2007/144097 A1, 2007 ;
Location in patent: Page/Page column 21 ;