1: SOCl2 / dimethylformamide / 0 - 20 °C
2: dimethylformamide / Ambient temperature
View Scheme
参考文献
Hamilton, Harriet W.; Ortwine, Daniel F.; Worth, Donald F.; Badger, Edward W.; Bristol, James A.; et al.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 8 p. 1071 - 1079
in N,N-dimethyl-formamide
Ambient temperature; Yield given;
参考文献
Hamilton, Harriet W.; Ortwine, Daniel F.; Worth, Donald F.; Badger, Edward W.; Bristol, James A.; et al.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 8 p. 1071 - 1079