4-(1-(4-硝基苯基)乙基)吗啉合成路线 (共 2 条)
反应条件
potassium carbonate in DMF (N,N-dimethyl-formamide)
T=20°C; 16 h;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2004/46120 A2, 2004 ;
Location in patent: Page 174 ;
WO 2004/046120 A2
反应条件
formic acid
T=100°C; 2 h;
参考文献
Nilsson, Asa; Carlson, Rolf
Acta Chemica Scandinavica, Series B: Organic Chemistry and Biochemistry, 1985 , vol. 39, # 3 p. 187 - 190