反应条件
1: 95 percent / pyridine; H2O / 18 h / 4 °C
2: 1.) n-BuLi, HMPA / 1.) THF, hexane, 20 min, 2.) THF, hexane, RT, 17 h
3: (Ph3P)3PdCl2, CuI, Et3N / 0.25 h
View Scheme
参考文献
Perchonock; Uzinskas; McCarthy; Erhard; Gleason; Wasserman; Muccitelli; DeVan; Tucker; Vickery
Journal of Medicinal Chemistry, 1986 , vol. 29, # 8 p. 1442 - 1452
