反应条件
1: 80 percent / triethylamine / CH2Cl2 / 2.5 h / -5 °C
2: 1.) Mg / 1.) THF, 2.) diglyme, 120-130 deg C, reflux 3h
View Scheme
参考文献
Buchowiecki, Wieslaw; Grosman-Zjawiona, Zofia; Zjawiony, Jordan
Tetrahedron Letters, 1985 , vol. 26, # 9 p. 1245 - 1248