反应条件
1: 100 percent / pyridine / CH2Cl2 / 1.) 0 deg C, 1 h, 2.) 25 deg C, overnight
2: 81 percent / BF3*Et2O / CH2Cl2 / 1.5 h / 0 °C
View Scheme
参考文献
Kassis, Pamela; Brzeszcz, Joanna; Beneteau, Valerie; Lozach, Olivier; Meijer, Laurent; Le Guevel, Remi; Guillouzo, Christiane; Lewinski, Krzysztof; Bourg, Stephane; Colliandre, Lionel; Routier, Sylvain; Merour, Jean-Yves
European Journal of Medicinal Chemistry, 2011 , vol. 46, # 11 p. 5416 - 5434