反应条件
1: 32 percent / aq. NaOH / dioxane / 0.5 h / 0 °C 2: aq. NaOH, Br2 / a) 0 deg C, 15 min, b) 90 deg C, 30 min View Scheme
参考文献
Egbertson, Melissa S.; Cook, Jacquelynn J.; Bednar, Bohumil; Prugh, John D.; Bednar, Rodney A.; Gaul, Stanley L.; Gould, Robert J.; Hartman, George D.; Homnick, Carl F.; Holahan, Marie A.; Libby, Laura A.; Lynch Jr., Joseph J.; Lynch, Robert J.; Sitko, Gary R.; Stranieri, Maria T.; Vassallo, Laura M.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 13 p. 2409 - 2421