1: With caesium carbonate; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl; palladium diacetate in toluene T=80°C; 2: With water; acetic acid in tetrahydrofuran
参考文献
Willis, Michael C.; Brace, Gareth N.
Tetrahedron Letters, 2002 , vol. 43, # 50 p. 9085 - 9088