1: pyridine / acetonitrile / 3 h / 0 - 10 °C 2: 22.94 kg / diisopropylethylamine / acetonitrile; ethyl acetate; H2O / 1 h / 10 - 20 °C View Scheme
参考文献
Farr, Roger N.; Alabaster, Ramon J.; Chung, John Y.L.; Craig, Bridgette; Edwards, John S.; Gibson, Andrew W.; Ho, Guo-Jie; Humphrey, Guy R.; Johnson, Simon A.; Grabowski
Tetrahedron Asymmetry, 2003 , vol. 14, # 22 p. 3503 - 3515