反应条件
1: 5-amino-2-sulfamoyl-1,3,4-thiadiazole monohydrochloride With triethylamine in dichloromethane
T=20°C; 1.5 h;
2: propionyl chloride in dichloromethane
T=20°C; 1.5 h;
参考文献
Schuettelkopf, Alexander W.; Gros, Ludovic; Blair, David E.; Frearson, Julie A.; Van Aalten, Daan M.F.; Gilbert, Ian H.
Bioorganic and Medicinal Chemistry, 2010 , vol. 18, # 23 p. 8334 - 8340
