1: 88 percent / Et3N / acetone / 24 h / 20 °C 2: 90 percent / DIEA; DMAP / dimethylformamide / 3 h / 20 °C 3: 98 percent / H2 / 10percent Pd/C / ethyl acetate / 1 h / 2280.15 Torr View Scheme
参考文献
August, Ryan A.; Khan, Jeffrey A.; Moody, Claire M.; Young, Douglas W.
Journal of the Chemical Society - Perkin Transactions 1, 1996 , # 6 p. 507 - 514