1-(4-溴苯甲酰基)哌啶合成路线 (共 12 条)
反应条件
1: PCl5
2: alkaline solution
View Scheme
参考文献
Schotten
Chemische Berichte, 1888 , vol. 21, p. 2251
反应条件
(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane; dichloromethane
T=80°C; 12 h;
参考文献
Patel, Gautam; Karver, Caitlin E.; Behera, Ranjan; Guyett, Paul J.; Sullenberger, Catherine; Edwards, Peter; Roncal, Norma E.; Mensa-Wilmot, Kojo; Pollastri, Michael P.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 10 p. 3820 - 3832