反应条件
1: potassium carbonate / N,N-dimethyl-formamide / 15 h / 20 °C
2: potassium carbonate; potassium iodide / N,N-dimethyl-formamide / 6 h / 80 °C
3: methanol; sodium hydroxide / 0.5 h / Reflux
View Scheme
参考文献
Levoin, Nicolas; Labeeuw, Olivier; Calmels, Thierry; Poupardin-Olivier, Olivia; Berrebi-Bertrand, Isabelle; Lecomte, Jeanne-Marie; Schwartz, Jean-Charles; Capet, Marc
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 18 p. 5378 - 5383