反应条件
1: potassium fluoride; kryptofix2.2.2; potassium carbonate / dimethylsulfoxide / 0.17 h / 150 °C 2: sodium hydroxide / dimethylsulfoxide; H2O / 0.08 h / 80 °C 3: 2.8 mg / hydrochloric acid; N-hydroxybenzotriazole; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide hydrochloride / H2O; dimethylformamide / 0.17 h / 20 °C View Scheme
参考文献
Murakami, Yoshihiro; Nishimura, Shintaro; Noda, Akihiro; Harada, Norihiro; Tsukada, Hideo
Journal of Labelled Compounds and Radiopharmaceuticals, 2002 , vol. 45, # 14 p. 1219 - 1228