反应条件
1: 30percent aq. H2O2 / acetic acid / 12 h / 80 °C 2: acetic anhydride / 1 h / Heating 3: 1.) NaH / 1.) DMF, 50 deg C, 0.5 h, 2.) DMF, 50 deg C, 2 h View Scheme
参考文献
Suzuki, Fumio; Kuroda, Takeshi; Nakasato, Yoshisuke; Manabe, Haruhiko; Ohmori, Kenji; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 22 p. 4045 - 4053