反应条件
1: 96 percent / K2CO3 / acetonitrile / 0.5 h / Heating
2: SO2Cl2, pyridine / 1.) RT, 0.5 h, 2.) 70 deg C, 4 h
View Scheme
参考文献
Watanabe, Nobuhisa; Kabasawa, Yasuhiro; Takase, Yasutaka; Matsukura, Masayuki; Miyazaki, Kazuki; Ishihara, Hiroki; Kodama, Kohtarou; Adachi, Hideyuki
Journal of Medicinal Chemistry, 1998 , vol. 41, # 18 p. 3367 - 3372