反应条件
1,8-diazabicyclo[5.4.0]undec-7-ene in acetonitrile
1.) reflux, 3 h, 2.) room temperature, 18 h;
参考文献
Sanchez, Joseph P.; Domagala, John M.; Hagen, Susan E.; Heifetz, Carl L.; Hutt, Marland P.; et al.
Journal of Medicinal Chemistry, 1988 , vol. 31, p. 983 - 991