甲基(2-氨基-1,3-苯并噻唑-6-基)乙酸酯合成路线 (共 1 条)
反应条件
1: With hydrogenchloride in 1,4-dioxane
T=75°C; 9 h;
2: With sodium hydroxide in water
pH=9;
参考文献
BRISTOL-MYERS SQUIBB COMPANY
Patent: WO2007/16392 A2, 2007 ;
Location in patent: Page/Page column 57 ;
WO 2007/016392 A2