反应条件
1: 54 percent / K2CO3 / dimethylsulfoxide / 4 h / Ambient temperature
2: 1.) BCl3, 2.) aq. NaOH / 1.) CH2Cl2, -78 deg C, 15 h, 2.) 80 deg C, 2 h
View Scheme
参考文献
Haines, David R.; Tseng, Christopher K. H.; Marquez, Victor E.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 5 p. 943 - 947