反应条件
sodium hydroxide; boron trichloride
1.) CH2Cl2, -78 deg C, 15 h, 2.) 80 deg C, 2 h; Yield given. Multistep reaction;
参考文献
Haines, David R.; Tseng, Christopher K. H.; Marquez, Victor E.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 5 p. 943 - 947